SCHEMBL27680337

SCHEMBL27680337

Brc1cc(-c2ccccc2)c[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.48
AURKB Q96GD4 2/20 0.48
MAPT P10636 2/20 0.48
THRB P10828 1/20 0.48
CASP1 P29466 1/20 0.48
TTK P33981 1/20 0.48
INCENP Q9NQS7 1/20 0.48
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
MCL1 Q07820 2/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 2/20 0.44
AKT1 P31749 1/20 0.41
AKT2 P31751 1/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
NOTUM Q6P988 1/20 0.39
IDO1 P14902 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14974312 0.74 AURKA (0.61) AURKAAURKBMAPTTHRBCASP1
SCHEMBL333740 0.73 MAPT (0.50) AURKAAURKBMAPTTHRBCASP1
SCHEMBL1126714 0.73 AURKA (0.50) AURKAAURKBMAPTTHRBCASP1
SCHEMBL24633981 0.73 ALDH1A1 (0.58) AURKAAURKBMAPTTHRBCASP1
SCHEMBL27844605 0.71 AURKA (0.48) AURKAAURKBMAPTTHRBCASP1
SCHEMBL6291849 0.71 MAPT (0.59) AURKAAURKBMAPTTHRBCASP1
SCHEMBL17279777 0.70 AURKA (0.47) AURKAAURKBMAPTTHRBCASP1
Biphenyl SCHEMBL4707139 0.69 ALDH1A1 (0.90) MAPTALDH1A1MAPK1AKT1AKT2
Biphenyl SCHEMBL5068276 0.69 ALDH1A1 (0.90) ALDH1A1MAPK1CRHBPCRHR2NOTUM
Perbromobenzene SCHEMBL28319870 0.67 ALDH1A1 (0.69) ALDH1A1MAPK1CRHBPCRHR2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106117181-A PI3K inhibitor and preparation method thereof and the application in pharmacy 复旦大学 2016-11-16 CN disclosed
CN-101027302-B Pyrrolo-pyridine kinase modulators SGX PHARMACEUTICALS INC 2011-05-11 CN disclosed
CN-101027302-A Pyrrolo-pyridine kinase modulators SGX PHARMACEUTICALS INC (US) 2007-08-29 CN disclosed