SCHEMBL27680360

SCHEMBL27680360

O=C(O)c1cccn1CCc1ccc(F)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.49
CA1 P00915 2/20 0.49
CA2 P00918 2/20 0.49
CA9 Q16790 2/20 0.49
CNR2 P34972 3/20 0.48
CNR1 P21554 2/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
FFAR1 O14842 1/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR7 P34969 1/20 0.40
HTR6 P50406 1/20 0.40
KDM5A P29375 1/20 0.40
KDM5B Q9UGL1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9023262 0.88 NPC1 (0.49) CNR2ALDH1A1
SCHEMBL20916882 0.86 NPC1 (0.51) KDM4EALDH1A1
SCHEMBL27680364 0.86 HDAC3 (0.51) KDM4EFFAR1
SCHEMBL1606703 0.83 CA12 (0.67) CA12CA1CA2CA9CNR2
SCHEMBL7177997 0.83 CA12 (0.46) CA12CA1CA2CA9CNR2
SCHEMBL28677395 0.83 FLT1 (0.42) CNR2CNR1KDM4E
SCHEMBL27680468 0.81 HTR2A (0.43) HTR2AHTR2C
SCHEMBL27660292 0.79 CCR2 (0.47)
SCHEMBL9023104 0.79 NPC1 (0.47) ALDH1A1
SCHEMBL27660326 0.79 ALDH1A1 (0.44) CA12CA1CA2CA9CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1922149-A Pyrrole and pyrazole daao inhibitors SEPRACOR INC (US) 2007-02-28 CN disclosed