SCHEMBL27681007

SCHEMBL27681007

NC(=O)c1cccnc1-c1cn[nH]c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.47
KDM4E B2RXH2 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
PIM1 P11309 2/20 0.41
RAB9A P51151 2/20 0.40
AKT1 P31749 1/20 0.40
AKT2 P31751 1/20 0.40
IKBKE Q14164 1/20 0.39
TBK1 Q9UHD2 1/20 0.39
PLK4 O00444 2/20 0.39
MAP4K4 O95819 2/20 0.39
FLT3 P36888 2/20 0.39
CSNK1A1 P48729 2/20 0.39
DYRK1B Q9Y463 2/20 0.39
CHEK1 O14757 1/20 0.39
AURKA O14965 1/20 0.39
DAPK3 O43293 1/20 0.39
CSF1R P07333 1/20 0.39
RET P07949 1/20 0.39
FGFR1 P11362 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30753661 0.86 KDM4E (0.61) KDM4ETDP1PIM1AKT1AKT2
SCHEMBL4186883 0.78 KDM4E (0.65) PARP1KDM4ETDP1RAB9ACSNK1A1
SCHEMBL22732136 0.78 PARP1 (0.43) PARP1KDM4ETDP1RAB9ACSNK1A1
SCHEMBL29916420 0.77 KDM4E (0.55) PARP1KDM4ETDP1RAB9ADYRK1B
SCHEMBL945856 0.77 KDM4E (0.55) PARP1KDM4ETDP1RAB9ADYRK1B
SCHEMBL4512695 0.76 BCAT2 (0.58) RAB9AAKT1AKT2PLK4MAP4K4
SCHEMBL1571384 0.76 MKNK1 (0.55) PARP1KDM4ETDP1MKNK2
SCHEMBL30387828 0.76 LRRK2 (0.38) PIM1AKT1AKT2IKBKETBK1
SCHEMBL29575496 0.76 MKNK1 (0.55) PARP1KDM4ETDP1MKNK2
SCHEMBL19520186 0.76 PARP1 (0.47) PARP1KDM4ETDP1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101023063-A Azine-carboxamides as anti-cancer agents ASTRAZENECA AB (SE) 2007-08-22 CN disclosed