SCHEMBL27683042

SCHEMBL27683042

COC(=O)N(C(=O)OC(C)(C)C)C(C)c1ccc(N)cc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALOX5 P09917 3/20 0.34
AAK1 Q2M2I8 2/20 0.34
CETP P11597 1/20 0.34
ADRB2 P07550 2/20 0.33
ADRB1 P08588 2/20 0.33
ADRB3 P13945 2/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28826276 0.88 ALOX5 (0.41) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL6762993 0.82 AAK1 (0.41) ALDH1A1NPC1MAPTMAPK1HTT
SCHEMBL17254362 0.79 ALOX5 (0.49) ALDH1A1NPC1MAPTRAB9AALOX5
SCHEMBL17241438 0.79 ALOX5 (0.49) ALDH1A1NPC1MAPTRAB9AALOX5
SCHEMBL17241382 0.78 MAPT (0.38) NPC1MAPTRAB9AL3MBTL1
SCHEMBL5780065 0.77 TYR (0.44) ALDH1A1NPC1MAPTRAB9AADRB2
SCHEMBL2953235 0.77 PTGS2 (0.47) ALOX5
SCHEMBL17254313 0.75 ALOX5 (0.33) ALOX5
SCHEMBL186630 0.72 ALOX5 (0.42) ALDH1A1L3MBTL1ALOX5
SCHEMBL3897727 0.72 ALOX5 (0.42) ALDH1A1L3MBTL1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100338036-C Substituted indolinones with inhibitory effect on kinase and cyclin complexes BOEHRINGER INGELHEIM PHARMA (DE) 2007-09-19 CN disclosed