SCHEMBL27684243

SCHEMBL27684243

C=C(c1ccc2c(c1)OCCO2)c1cn(S(=O)(=O)O)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.40
CTNNB1 P35222 5/20 0.39
HPGD P15428 3/20 0.39
RECQL P46063 1/20 0.39
WNT3A P56704 3/20 0.38
KDM4E B2RXH2 2/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 4/20 0.38
RAB9A P51151 4/20 0.38
CTSZ Q9UBR2 2/20 0.38
GAA P10253 1/20 0.38
HTT P42858 1/20 0.38
NPC1 O15118 3/20 0.38
TP53 P04637 2/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PKM P14618 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3751611 0.86 POLB (0.42) TSHRCTNNB1HPGDKDM4EATM
SCHEMBL13081422 0.80 TSHR (0.41) TSHRCTNNB1HPGDRECQLWNT3A
SCHEMBL7453623 0.64 TSHR (0.54) TSHRCTNNB1HPGDRECQLKDM4E
SCHEMBL2496047 0.62 TSHR (0.72) TSHRCTNNB1HPGDRECQLWNT3A
SCHEMBL16071127 0.62 TSHR (0.56) TSHRCTNNB1HPGDRECQLWNT3A
SCHEMBL28530741 0.62 TSHR (0.61) TSHRCTNNB1HPGDRECQLKDM4E
SCHEMBL4824992 0.62 NPSR1 (0.74) TSHRCTNNB1HPGDRECQLWNT3A
Formaldehyde SCHEMBL27289523 0.61 MAPK1 (0.72) TSHRCTNNB1HPGDRECQLKDM4E
SCHEMBL619634 0.61 MAPK1 (0.78) TSHRCTNNB1HPGDRECQLKDM4E
SCHEMBL16795707 0.60 TSHR (0.53) TSHRCTNNB1HPGDRECQLWNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101052638-B As α24- (condensed cyclomethyl) -imidazole-2-thiones as adrenergic agonists ALLERGAN INC 2011-01-19 CN disclosed
CN-101052638-A As α24- (condensed cyclomethyl) adrenergic agonists-imidazole-2-thiones ALLERGAN INC (US) 2007-10-10 CN disclosed