SCHEMBL27686153

SCHEMBL27686153

CNc1cc(-c2ccc(F)cc2)cnc1OC(C)=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 4/20 0.47
MAP4K4 O95819 1/20 0.41
GRIN2B Q13224 4/20 0.39
GRIN1 Q05586 1/20 0.39
IKBKB O14920 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
HDAC1 Q13547 2/20 0.38
FYN P06241 1/20 0.38
HDAC2 Q92769 1/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
SCN10A Q9Y5Y9 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28765654 0.82 CYP4F2 (0.39) CHRNA7NPC1RAB9ASMN1; SMN2
SCHEMBL27667112 0.81 MAPT (0.47) CHRNA7MAP4K4GRIN2BGRIN1IKBKB
SCHEMBL27686155 0.77 CHRNA7 (0.46) CHRNA7GRIN2BGRIN1IKBKBEGLN1
SCHEMBL27686102 0.76 MAPT (0.39) CHRNA7MAP4K4GRIN2BGRIN1PDGFRB
SCHEMBL28765670 0.69 CYP11B1 (0.41)
SCHEMBL28736437 0.68 MAP4K4 (0.47) CHRNA7MAP4K4GRIN2BGRIN1IKBKB
SCHEMBL22083773 0.67 HSD17B10 (0.63) RAB9ASMN1; SMN2
SCHEMBL4940831 0.66 SSTR4 (0.40) HDAC1HDAC2PIK3CA
SCHEMBL28772992 0.66 CYP17A1 (0.40) MAP4K4FYNNPC1RAB9ASMN1; SMN2
SCHEMBL27803399 0.66 PTGS1 (0.41) NPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed