SCHEMBL27686155

SCHEMBL27686155

CNc1cc(-c2ccc(F)cc2)cnc1C(=O)OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.46
EGLN1 Q9GZT9 1/20 0.45
GRIN2B Q13224 5/20 0.42
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
NPC1 O15118 1/20 0.41
CASP3 P42574 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SENP8 Q96LD8 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
ACLY P53396 1/20 0.41
IKBKB O14920 2/20 0.40
GRIN1 Q05586 1/20 0.40
MAP2K4 P45985 1/20 0.40
DHODH Q02127 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27667113 0.82 IKBKB (0.50) CHRNA7EGLN1GRIN2BPDGFRBPDGFRA
SCHEMBL5547230 0.81 MAPT (0.41) NPC1RAB9ASMN1; SMN2
SCHEMBL23484278 0.78 CHRNA7 (0.49) CHRNA7EGLN1GRIN2BPDGFRBPDGFRA
SCHEMBL27686103 0.78 ERN1 (0.44) EGLN1GRIN2BPDGFRBPDGFRASLC6A4
SCHEMBL27686153 0.77 CHRNA7 (0.47) CHRNA7EGLN1GRIN2BPDGFRBPDGFRA
SCHEMBL16634586 0.75 SLC6A4 (0.51) EGLN1SLC6A4SLC6A3NPC1CASP3
SCHEMBL22116633 0.73 NPSR1 (0.39) SMN1; SMN2LMNA
SCHEMBL2906199 0.71 CYP11B1 (0.62) NPC1RAB9AMAP2K4
SCHEMBL4715889 0.70 MEN1 (0.41) NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL5004713 0.70 LMNA (0.44) NPC1CASP3RAB9ASMN1; SMN2SENP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed