SCHEMBL27686339

SCHEMBL27686339

NC(=O)c1c(C(Cc2ncc[nH]2)C(O)N2CCOCC2)c2ncc(Cc3ccc(F)cc3)cc2[nH]c1=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.33
NAMPT P43490 2/20 0.32
XIAP P98170 1/20 0.31
BIRC2 Q13490 1/20 0.31
HTR2B P41595 1/20 0.31
GRM2 Q14416 1/20 0.31
PIK3CD O00329 2/20 0.31
PIK3CB P42338 2/20 0.31
PARP1 P09874 1/20 0.31
STAT6 P42226 1/20 0.30
AKT1 P31749 2/20 0.30
HSD17B10 Q99714 1/20 0.30
AURKA O14965 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
CDK2 P24941 1/20 0.30
AURKB Q96GD4 1/20 0.30
CYP3A4 P08684 1/20 0.30
PIK3CA P42336 1/20 0.30
GRIN2B Q13224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27667070 0.84 NTRK1 (0.36) NTRK1XIAPBIRC2GRM2PARP1
SCHEMBL27666972 0.81 NTRK1 (0.36) NTRK1XIAPBIRC2GRM2PARP1
SCHEMBL27686180 0.77 GRM2 (0.34) GRM2
SCHEMBL27667063 0.74 GRM2 (0.34) XIAPBIRC2GRM2PARP1
SCHEMBL27666982 0.72 BTK (0.34) GRM2PARP1HSD17B10
SCHEMBL5546423 0.71 TDP1 (0.40) GRM2HSD17B10GRIN2B
SCHEMBL27667075 0.70 GRM2 (0.33) GRM2
SCHEMBL27667206 0.70 SCN9A (0.36) GRM2
SCHEMBL5539022 0.69 NTRK1 (0.39) NTRK1XIAPBIRC2PARP1AURKA
SCHEMBL27667170 0.69 BTK (0.33) GRM2PARP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed