SCHEMBL27666972

SCHEMBL27666972

NC(=O)c1c(CC(O)N2CCOCC2)c2ncc(Cc3ccc(F)cc3)cc2[nH]c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.36
GRM2 Q14416 3/20 0.34
XIAP P98170 3/20 0.34
BIRC2 Q13490 3/20 0.34
GRIN2B Q13224 2/20 0.33
HTR2C P28335 1/20 0.33
MCHR1 Q99705 1/20 0.33
PARP1 P09874 6/20 0.33
PARP2 Q9UGN5 2/20 0.33
TNKS O95271 1/20 0.33
PARP6 Q2NL67 1/20 0.33
PARP3 Q9Y6F1 1/20 0.33
KCNH2 Q12809 2/20 0.33
NR1I2 O75469 1/20 0.33
STAT6 P42226 1/20 0.32
HSD17B10 Q99714 2/20 0.32
GAA P10253 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27667166 0.88 NTRK1 (0.32) NTRK1XIAPGRIN2BHTR2CMCHR1
SCHEMBL27667070 0.85 NTRK1 (0.36) NTRK1GRM2XIAPBIRC2GRIN2B
SCHEMBL27666982 0.85 BTK (0.34) GRM2PARP1PARP2TNKSPARP6
SCHEMBL27667206 0.82 SCN9A (0.36) GRM2
SCHEMBL27686339 0.81 NTRK1 (0.33) NTRK1GRM2XIAPBIRC2GRIN2B
SCHEMBL27686061 0.81 TDP1 (0.36) GRM2PARP1PARP2TNKSPARP6
SCHEMBL28767160 0.81 GRM2 (0.35) GRM2KCNH2MAPK1
SCHEMBL27667170 0.80 BTK (0.33) GRM2PARP1PARP2TNKSPARP6
SCHEMBL27667135 0.80 GRIN2B (0.42) NTRK1GRIN2BALDH1A1SMN1; SMN2
SCHEMBL27686178 0.79 PIK3CA (0.39) NTRK1GRM2GRIN2BHTR2CMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN claimed
CN-1976915-A HIV integrase inhibitors SMITHKLINE BEECHAM CORP (US) 2007-06-06 CN disclosed