SCHEMBL27687489

SCHEMBL27687489

C#Cc1cc(-c2ccncc2)sc1-c1nc2cnccn2c1NCCCC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.49
CDK9 P50750 1/20 0.43
ATM Q13315 5/20 0.43
APAF1 O14727 1/20 0.43
TLR9 Q9NR96 2/20 0.42
IDE P14735 1/20 0.41
PLAU P00749 1/20 0.40
GAA P10253 4/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
CASP1 P29466 2/20 0.38
CASP7 P55210 2/20 0.38
HSD17B10 Q99714 2/20 0.38
TRIM33 Q9UPN9 2/20 0.37
ALOX15 P16050 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27687439 0.92 BRD4 (0.48) BRD4CDK9ATMAPAF1TLR9
SCHEMBL5128033 0.81 BRD4 (0.48) BRD4CDK9ATMAPAF1TLR9
SCHEMBL5113401 0.81 BRD4 (0.53) BRD4CDK9ATMAPAF1TLR9
SCHEMBL5122857 0.79 BRD4 (0.45) BRD4CDK9ATMAPAF1TLR9
SCHEMBL27706739 0.78 BRD4 (0.52) BRD4CDK9ATMAPAF1TLR9
SCHEMBL5129311 0.76 PLAU (0.42) BRD4CDK9ATMAPAF1TLR9
SCHEMBL27687440 0.76 ALDH1A1 (0.42) ATMALDH1A1TRIM33NPC1RAB9A
SCHEMBL27687488 0.73 BRD4 (0.49) BRD4CDK9ATMAPAF1TLR9
SCHEMBL7980039 0.73 BRD4 (0.67) BRD4CDK9ATMAPAF1TLR9
SCHEMBL6642431 0.72 BRD4 (0.56) BRD4CDK9ATMAPAF1TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101061118-A Substituted bicyclic imidazo-3-ylamine compounds GRUENENTHAL GMBH (DE) 2007-10-24 CN disclosed