SCHEMBL7980039

SCHEMBL7980039

CCCCNc1c(-c2ccccc2)nc2cnccn12

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.67
CDK9 P50750 1/20 0.62
ATM Q13315 6/20 0.60
APAF1 O14727 1/20 0.60
GAA P10253 5/20 0.59
KDM4E B2RXH2 3/20 0.59
LMNA P02545 1/20 0.59
MAPK1 P28482 1/20 0.59
TLR9 Q9NR96 2/20 0.58
BRAF P15056 2/20 0.56
IDE P14735 1/20 0.52
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
ALDH1A1 P00352 2/20 0.50
HPGD P15428 2/20 0.50
CASP1 P29466 2/20 0.50
CASP7 P55210 2/20 0.50
HSD17B10 Q99714 2/20 0.50
ALOX15 P16050 1/20 0.50
TP53 P04637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6747493 0.85 ATM (0.65) BRD4ATMGAAKDM4ENPC1
SCHEMBL27528806 0.83 GAA (0.60) BRD4ATMAPAF1GAAKDM4E
SCHEMBL5880576 0.81 CDK9 (0.90) BRD4CDK9GAAKDM4ELMNA
SCHEMBL16416734 0.81 BRD4 (1.00) BRD4ATMAPAF1GAAKDM4E
SCHEMBL5166866 0.81 PKM (0.64) BRD4ATMGAAKDM4ELMNA
SCHEMBL6642431 0.80 BRD4 (0.56) BRD4CDK9ATMAPAF1GAA
SCHEMBL5167573 0.80 BRD4 (0.51) BRD4CDK9ATMAPAF1GAA
SCHEMBL5113389 0.79 BRD4 (0.48) BRD4CDK9ATMAPAF1GAA
SCHEMBL5128028 0.79 BRD4 (0.48) BRD4CDK9ATMAPAF1GAA
SCHEMBL31193263 0.79 CDK9 (0.60) BRD4CDK9ATMAPAF1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001027119-A2 SUBSTANCE LIBRARY CONTAINING BICYCLIC IMIDAZO-5-YL-AMINES AND/OR BICYCLIC IMIDAZO-3-YL-AMINES Grünenthal GmbH (DE) 2001-04-19 WO claimed
WO-2001027119-A2 SUBSTANCE LIBRARY CONTAINING BICYCLIC IMIDAZO-5-YL-AMINES AND/OR BICYCLIC IMIDAZO-3-YL-AMINES Grünenthal GmbH (DE) 2001-04-19 WO disclosed