SCHEMBL276887

SCHEMBL276887

CCCCCCCC(CC)OC(C)=O

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PRKCA P17252 3/20 0.50
GLS2 Q9UI32 3/20 0.49
FAAH O00519 2/20 0.45
PRKCD Q05655 1/20 0.44
GPR84 Q9NQS5 3/20 0.44
FFAR1 O14842 1/20 0.44
MAPT P10636 2/20 0.43
ZDHHC7 Q9NXF8 1/20 0.43
MAPK1 P28482 1/20 0.43
LCK P06239 1/20 0.42
PPARD Q03181 1/20 0.42
ZDHHC20 Q5W0Z9 1/20 0.42
ZDHHC2 Q9UIJ5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28751563 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL30731537 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL29655357 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL31626952 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL2486538 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL23930714 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL227644 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL19971880 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL22471650 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84
SCHEMBL27642486 1.00 PRKCA (0.50) PRKCAGLS2FAAHPRKCDGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4585893-A Process for producing 4-homoisotwistane-3-carboxylic acid KAO CORPORATION (JP) 1986-04-29 US claimed
US-11891642-B2 Biocatalytic techniques HYPHA DISCOVERY LIMITED (GB) 2024-02-06 US disclosed
CN-111527090-B Pyrazolo-pyrrolo-pyrimidine-dione derivatives as P2X3 inhibitors 拜耳公司 2023-05-26 CN disclosed
US-20220025416-A1 BIOCATALYTIC TECHNIQUES HYPHA DISCOVERY LIMITED (GB) 2022-01-27 US disclosed
EP-3887512-A2 BIOCATALYTIC TECHNIQUES Hypha Discovery Ltd. (GB) 2021-10-06 EP disclosed
CN-111527090-A Novel pyrazolo-pyrrolo-pyrimidine-dione derivatives as P2X3 inhibitors 拜耳公司 2020-08-11 CN disclosed
WO-2020109776-A2 BIOCATALYTIC TECHNIQUES HYPHA DISCOVERY LIMITED (GB) 2020-06-04 WO disclosed
CN-110650738-A Compounds and methods for treating parasitic diseases 博德研究所 2020-01-03 CN disclosed
US-10408819-B2 Luminescence-based methods and probes for measuring cytochrome P450 activity PROMEGA CORPORATION (US) 2019-09-10 US disclosed
US-20170191985-A1 LUMINESCENCE-BASED METHODS AND PROBES FOR MEASURING CYTOCHROME P450 ACTIVITY JPMORGAN CHASE BANK, N.A., AS COLLATERAL AGENT 2017-07-06 US disclosed
WO-2004027378-A2 LUMINESCENCE-BASED METHODS AND PROBES FOR MEASURING CYTOCHROME P450 ACTIVITY PROMEGA CORPORATION (US) 2004-04-01 WO disclosed
EP-1183252-B1 PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2004-02-18 EP disclosed
US-6492406-B1 PROTEIN KINASE C INHIBITORS; ANTIINFLAMMATORY AND IMMUNO-SUPPRESSIVE AGENTS ASTRAZENECA AB (SE) 2002-12-10 US disclosed
EP-1183252-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2002-03-06 EP disclosed
WO-2000071537-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 2000-11-30 WO disclosed
US-5270334-A 4-methoxy-5-methyl-pyran-3-ol natural products and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1993-12-14 US disclosed
US-5248790-A Antibiotics E. R. SQUIBB & SONS, INC. (US) 1993-09-28 US disclosed
US-4226903-A PAPER, ARAMIDS, THERMOSETTING RESINS GENERAL ELECTRIC COMPANY (US) 1980-10-07 US disclosed
US-4171969-A Bis(aminomethyl)phosphinic acid CIBA-GEIGY CORPORATION (US) 1979-10-23 US disclosed
US-4163912-A Electrical insulating sheet material and electric winding made therefrom GENERAL ELECTRIC COMPANY (US) 1979-08-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10408819-B2 Luminescence-based methods and probes for measuring cytochrome P450 activity CYP3A7, CYP3A43, CYP3A5 PRKCA 4476/4885GLS2 49/4885FAAH 1183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.