SCHEMBL27697668

SCHEMBL27697668

Cc1ccc(C(C)C(=O)C(C)c2ccc(C)cc2O)c(O)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.64
LMNA P02545 2/20 0.64
CHRM1 P11229 1/20 0.64
SLC6A2 P23975 1/20 0.64
ADRA1A P35348 1/20 0.64
HTR2B P41595 1/20 0.64
SRC P12931 1/20 0.46
CSNK2A1 P68400 1/20 0.42
ALDH1A1 P00352 3/20 0.42
GAA P10253 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
TP53 P04637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11064558 0.86 TRPA1 (0.62) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL28238190 0.86 TRPA1 (0.62) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL27536509 0.82 TYR (0.52) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL27766136 0.82 TRPA1 (0.45) TRPA1LMNACHRM1SLC6A2ADRA1A
Thymol SCHEMBL28150359 0.80 TRPA1 (0.84) TRPA1LMNACHRM1SLC6A2ADRA1A
Sulfuric Acid SCHEMBL11109027 0.79 LMNA (0.53) TRPA1LMNACHRM1SLC6A2ADRA1A
Thymol SCHEMBL22165 0.79 LMNA (1.00) TRPA1LMNACHRM1SLC6A2ADRA1A
SCHEMBL51957 0.79 LMNA (0.75) TRPA1LMNACHRM1SLC6A2ADRA1A
Thymol SCHEMBL29579824 0.79 LMNA (1.00) TRPA1LMNACHRM1SLC6A2ADRA1A
Thymol SCHEMBL30332213 0.79 LMNA (1.00) TRPA1LMNACHRM1SLC6A2ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105330675-A Inhibitors of HIV replication VIIV HEAL THCARE UK LTD 2016-02-17 CN disclosed
CN-103429595-B Inhibitors of HIV Replication VIIV HEALTHCARE UK LTD. (GB) 2015-10-21 CN disclosed
CN-103429595-A Inhibitors of hiv replication VIIV HEALTHCARE UK LTD 2013-12-04 CN disclosed
CN-101855224-B Equilibrative nucleoside transporter ENT1 inhibitors JANSSEN PHARMACEUTICA NV 2012-11-28 CN disclosed
CN-101855224-A Equilibrative nucleoside transporter ENT 1 inhibitors JANSSEN PHARMACEUTICA NV 2010-10-06 CN disclosed
CN-101146798-A Novel heterocyclic benzo[C]chromene derivatives useful as modulators of the estrogen receptors JANSSEN PHARMACEUTICA NV (BE) 2008-03-19 CN disclosed