SCHEMBL27699210

SCHEMBL27699210

FC(F)(F)c1cccc(-c2cn(-c3cccnc3)cn2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 1/20 0.49
CYP2E1 P05181 2/20 0.49
CYP2A6 P11509 2/20 0.49
PIM1 P11309 1/20 0.47
KCNA5 P22460 2/20 0.44
IDO1 P14902 1/20 0.44
KIF11 P52732 1/20 0.44
GRIN2B Q13224 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
GRIN1 Q05586 2/20 0.43
POLB P06746 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAOB P27338 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
NLRP3 Q96P20 1/20 0.42
MC4R P32245 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27699234 0.83 CYP2A6 (0.52) CYP2E1CYP2A6PIM1IDO1GRIN2B
SCHEMBL27699427 0.81 CYP2A6 (0.59) CYP2E1CYP2A6ALDH1A1CYP2C9CYP2B6
SCHEMBL27719699 0.80 CYP2A6 (0.52) NPY5RCYP2E1CYP2A6KCNA5IDO1
SCHEMBL27719703 0.80 MEN1 (0.54) CYP2E1CYP2A6ALDH1A1POLBCYP2C9
SCHEMBL16658968 0.79 KEAP1 (0.58) NPY5RPIM1
SCHEMBL27719702 0.77 GRM5 (0.56) CYP2E1CYP2A6IDO1ALDH1A1CYP2C19
SCHEMBL27812074 0.77 KMO (0.59) CYP2E1CYP2A6ALDH1A1CYP2C9CYP2B6
SCHEMBL15825417 0.77 CYP2A6 (0.55) CYP2E1CYP2A6CYP2C9CYP2B6CYP2C19
SCHEMBL27832179 0.76 HSP90AA1 (0.52) CYP2E1CYP2A6PIM1
SCHEMBL12710038 0.75 MEN1 (0.63) NPY5RPIM1KCNA5KIF11GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101166735-A Novel oxadiazole derivatives and their medical use NEUROSEARCH AS (DK) 2008-04-23 CN claimed
CN-101166735-A Novel oxadiazole derivatives and their medical use NEUROSEARCH AS (DK) 2008-04-23 CN disclosed