SCHEMBL2769939

SCHEMBL2769939

Cc1cc(OCc2c(C(C)C)cnn2-c2ccccc2OC(F)(F)F)ccc1C(C)(C)Sc1ccc(C(=O)O)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.41
RXRA P19793 2/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
LNPEP Q9UIQ6 1/20 0.34
P2RY1 P47900 1/20 0.33
HSD17B13 Q7Z5P4 1/20 0.32
PPARD Q03181 4/20 0.32
PPARA Q07869 2/20 0.32
MRGPRX4 Q96LA9 2/20 0.31
HNF4A P41235 1/20 0.31
TRPM8 Q7Z2W7 2/20 0.31
GLP1R P43220 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2771301 0.93 NR1H4 (0.43) NR1H4LNPEPP2RY1PPARDPPARA
SCHEMBL2771573 0.92 NR1H4 (0.40) NR1H4LNPEPP2RY1PPARDPPARA
SCHEMBL2775274 0.88 NR1H4 (0.40) NR1H4LNPEPP2RY1PPARDPPARA
SCHEMBL2770877 0.85 NR1H4 (0.42) NR1H4RXRARXRBRXRGLNPEP
SCHEMBL2771604 0.83 NR1H4 (0.59) NR1H4MRGPRX4
SCHEMBL2773384 0.83 TRPM8 (0.40) NR1H4RXRARXRBRXRGPPARA
SCHEMBL2769947 0.82 NR1H4 (0.39) NR1H4RXRARXRBRXRGLNPEP
SCHEMBL2770116 0.81 KDM4E (0.40) NR1H4RXRARXRBRXRGLNPEP
SCHEMBL2771175 0.81 NR1H4 (0.44) NR1H4LNPEPPPARDMRGPRX4
SCHEMBL2770864 0.80 NR1H4 (0.39) NR1H4LNPEPP2RY1PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed