SCHEMBL2770877

SCHEMBL2770877

Cc1cc(OCc2c(C(C)C)cnn2-c2ccccc2OC(F)(F)F)ccc1-c1ccc(C(=O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.42
HSD17B13 Q7Z5P4 1/20 0.39
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
LNPEP Q9UIQ6 1/20 0.38
PPARD Q03181 7/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 2/20 0.36
NTRK1 P04629 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
MAP4K4 O95819 1/20 0.35
CETP P11597 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2770866 0.89 NR1H4 (0.43) NR1H4RXRARXRBRXRGPPARD
SCHEMBL2773384 0.86 TRPM8 (0.40) NR1H4RXRARXRBRXRGPPARA
SCHEMBL2770076 0.86 NR1H4 (0.51) NR1H4
SCHEMBL2773202 0.86 PPARD (0.36) NR1H4LNPEPPPARDPPARA
SCHEMBL3149710 0.86 NR1H4 (0.46) NR1H4HSD17B13RXRARXRBRXRG
SCHEMBL2770752 0.86 NR1H4 (0.39) NR1H4LNPEPPPARDPPARG
SCHEMBL2770864 0.85 NR1H4 (0.39) NR1H4LNPEPPPARDFFAR4
SCHEMBL2770116 0.85 KDM4E (0.40) NR1H4RXRARXRBRXRGLNPEP
SCHEMBL2769939 0.85 NR1H4 (0.41) NR1H4HSD17B13RXRARXRBRXRG
SCHEMBL2769947 0.85 NR1H4 (0.39) NR1H4RXRARXRBRXRGLNPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed