SCHEMBL27699501

SCHEMBL27699501

NC(=O)C1CC1c1ccc(C(F)(F)F)nc1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.58
HDAC4 P56524 1/20 0.44
KCNH2 Q12809 1/20 0.43
CYP3A4 P08684 1/20 0.40
NAMPT P43490 1/20 0.40
FFAR1 O14842 1/20 0.39
KDM1A O60341 4/20 0.39
MAOB P27338 3/20 0.39
TRPV4 Q9HBA0 1/20 0.39
SLC9A1 P19634 1/20 0.38
MAOA P21397 2/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA4 P43681 1/20 0.38
CHRNA7 P36544 1/20 0.38
FAAH O00519 1/20 0.38
DGAT1 O75907 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27813823 0.88 HRH3 (0.60) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL451176 0.87 HRH3 (0.59) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL451175 0.87 HRH3 (0.59) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL15314478 0.87 HRH3 (0.59) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL12128175 0.87 HRH3 (0.59) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL23550031 0.85 HRH3 (0.58) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL18529756 0.85 HRH3 (0.44) HRH3KCNH2CYP3A4NAMPTFFAR1
SCHEMBL12128172 0.82 HRH3 (0.55) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL451266 0.82 HRH3 (0.55) HRH3HDAC4KCNH2CYP3A4NAMPT
SCHEMBL15314513 0.82 HRH3 (0.55) HRH3HDAC4KCNH2CYP3A4NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101160285-A Substituted sulfonylaminoarylmethyl cyclopropanecarboxamide as vr1 receptor antagonists PFIZER (US) 2008-04-09 CN disclosed