SCHEMBL27699861

SCHEMBL27699861

CC(Br)c1c(-c2ccc(F)cc2)c2ccccc2oc1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.48
MAPK14 Q16539 2/20 0.46
GABRP O00591 1/20 0.46
GABRD O14764 1/20 0.46
TNKS O95271 1/20 0.46
PARP1 P09874 1/20 0.46
GABRA1 P14867 1/20 0.46
GABRB1 P18505 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
GABRA2 P47869 1/20 0.46
GABRB2 P47870 1/20 0.46
GABRA4 P48169 1/20 0.46
GABRE P78334 1/20 0.46
GABRA6 Q16445 1/20 0.46
GABRG1 Q8N1C3 1/20 0.46
GABRG3 Q99928 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18150081 0.89 VKORC1 (0.50) VKORC1MGAMGAASIMGAM2
SCHEMBL8552 0.80 MAPK14 (0.53) PTGS2MAPK14GABRPGABRDTNKS
SCHEMBL31511408 0.77 TNKS (0.53) PTGS2MAPK14GABRPGABRDTNKS
SCHEMBL18150266 0.74 VKORC1 (0.54) VKORC1ALDH1A1NQO1CYP2C9CRHBP
SCHEMBL27699860 0.73 NPC1 (0.48) PTGS2MAPK14GABRPGABRDTNKS
SCHEMBL8336100 0.73 VKORC1 (0.74) VKORC1TOP2AALDH1A1NQO1CYP2C9
SCHEMBL11480111 0.73 MAOB (0.68) PTGS2MAPK14GABRPGABRDTNKS
SCHEMBL9011 0.71 MAPK14 (0.50) PTGS2MAPK14GABRPGABRDTNKS
SCHEMBL8364 0.71 MAPK14 (0.59) PTGS2MAPK14GABRPGABRDTNKS
SCHEMBL28582663 0.70 GABRP (0.49) PTGS2MAPK14GABRPGABRDTNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101146802-A Thiadiazole-substituted coumarin derivatives and their use as leukotriene biosynthesis inhibitors MERCK FROSST CANADA LTD (CA) 2008-03-19 CN disclosed