SCHEMBL27701503

SCHEMBL27701503

NC(=O)c1ccc(Cc2cccnc2)c(C(N)=O)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.46
GRM2 Q14416 1/20 0.44
TBXAS1 P24557 7/20 0.43
NAPRT Q6XQN6 1/20 0.43
PNP P00491 1/20 0.43
CYP3A4 P08684 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
F7 P08709 1/20 0.41
F3 P13726 1/20 0.41
SARM1 Q6SZW1 1/20 0.41
SIRT2 Q8IXJ6 1/20 0.41
SIRT6 Q8N6T7 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41
SIRT5 Q9NXA8 1/20 0.41
SIRT4 Q9Y6E7 1/20 0.41
MEN1 O00255 1/20 0.41
TP53 P04637 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28613561 0.84 PLA2G10 (0.46) MEN1KMT2A
SCHEMBL13728047 0.76 GRM2 (0.47) RECQLGRM2TBXAS1NAPRTCYP3A4
SCHEMBL29817984 0.74 RECQL (0.50) RECQLTBXAS1NAPRTCYP3A4CYP1A2
SCHEMBL16598255 0.74 RECQL (0.50) RECQLTBXAS1NAPRTCYP3A4CYP1A2
SCHEMBL28826508 0.74 IKBKB (0.54) CYP3A4CYP1A2F7F3SARM1
SCHEMBL1161996 0.74 RECQL (0.50) RECQLTBXAS1NAPRTCYP3A4CYP1A2
Hydrochloric Acid SCHEMBL17906582 0.72 RECQL (0.49) RECQLTBXAS1NAPRTCYP3A4CYP1A2
SCHEMBL28190937 0.72 TBXAS1 (0.46) RECQLTBXAS1NAPRTCYP3A4CYP1A2
Hydrochloric Acid SCHEMBL17204692 0.71 RECQL (0.44) RECQLGRM2TBXAS1NAPRTCYP3A4
SCHEMBL13728559 0.71 RECQL (0.44) RECQLGRM2TBXAS1NAPRTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101014571-A N-benzyl-3,4-dihyroxypyridine-2-carboxamide and n-benzyl-2,3-dihydroxypyridine-4- carboxamide compounds useful as HIV integrase inhibitors MERCK & CO INC (US) 2007-08-08 CN disclosed