SCHEMBL27701893

SCHEMBL27701893

Cc1nc(Cl)c(N2CCNCC2)c(Cc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 2/20 0.47
TAAR1 Q96RJ0 1/20 0.47
HTR6 P50406 3/20 0.45
SOS1 Q07889 1/20 0.44
HTR3A P46098 1/20 0.42
ADRB1 P08588 1/20 0.42
NCF1 P14598 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
HTR2C P28335 2/20 0.41
HTR2A P28223 1/20 0.41
HTR2B P41595 1/20 0.41
PIM1 P11309 1/20 0.40
PDE10A Q9Y233 1/20 0.40
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27702067 0.86 HRH4 (0.47) CETPTAAR1HTR6HTR3AADRB1
SCHEMBL27701890 0.85 CETP (0.49) CETPTAAR1HTR6HTR3ASIGMAR1
SCHEMBL27701987 0.82 POLB (0.54) CETPTAAR1HTR6HTR3AHTR2C
SCHEMBL27682791 0.73 CETP (0.58) CETPTAAR1HTR6HTR2CHTR2A
SCHEMBL1830467 0.70 SMO (0.70) TAAR1HTR2CHPGD
SCHEMBL10078401 0.69 TAAR1 (0.50) CETPTAAR1HTR6HTR3AADRB1
SCHEMBL21794745 0.69 TAAR1 (0.44) CETPTAAR1HTR6SOS1HTR3A
SCHEMBL5788785 0.68 ALDH1A1 (0.60) CETPTAAR1HTR6HTR3AADRB1
SCHEMBL27737301 0.68 CETP (0.58) CETPTAAR1HTR6HTR3AHTR2C
SCHEMBL20315055 0.68 MEN1 (0.58) TAAR1CYP1A2CYP3A4HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101054372-B Pyrimidine substituted benzenepropanoic acid derivative, its preparation method and use in curing polycystic kidney disease SHANGHAI INST MATERIA MEDICA 2010-10-13 CN disclosed
CN-101054372-A Pyrimidine substituted benzenepropanoic acid derivative, its preparation method and use in curing polycystic kidney disease SHANGHAI INST MATERIA MEDICA (CN) 2007-10-17 CN disclosed