SCHEMBL27701987

SCHEMBL27701987

Clc1nc(Nc2ccccc2)nc(Cc2ccccc2)c1N1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.54
KMT2A Q03164 1/20 0.54
ALDH1A1 P00352 2/20 0.50
ROCK1 Q13464 3/20 0.48
CETP P11597 2/20 0.43
TAAR1 Q96RJ0 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
HTR2A P28223 2/20 0.40
LMNA P02545 1/20 0.39
HTR6 P50406 2/20 0.39
KDM1A O60341 1/20 0.39
HTR3A P46098 1/20 0.39
STAT6 P42226 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27701893 0.82 CETP (0.47) ALDH1A1CETPTAAR1HTR2AHTR6
SCHEMBL27702067 0.81 HRH4 (0.47) CETPTAAR1HTR2AHTR6HTR3A
SCHEMBL27701890 0.80 CETP (0.49) KMT2AALDH1A1CETPTAAR1HTR2A
SCHEMBL15613209 0.71 POLB (1.00) POLBKMT2AALDH1A1ROCK1TAAR1
SCHEMBL27617368 0.70 POLB (0.84) POLBKMT2AALDH1A1ROCK1CETP
SCHEMBL27682791 0.68 CETP (0.58) POLBKMT2ACETPTAAR1HTR2A
SCHEMBL15613241 0.68 ALDH1A1 (0.97) POLBKMT2AALDH1A1ROCK1TAAR1
SCHEMBL16872901 0.67 ALDH1A1 (1.00) POLBKMT2AALDH1A1ROCK1TAAR1
SCHEMBL27598825 0.66 POLB (0.86) POLBKMT2AALDH1A1ROCK1TAAR1
SCHEMBL15800688 0.66 POLB (0.74) POLBKMT2AALDH1A1ROCK1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101054372-B Pyrimidine substituted benzenepropanoic acid derivative, its preparation method and use in curing polycystic kidney disease SHANGHAI INST MATERIA MEDICA 2010-10-13 CN disclosed
CN-101054372-A Pyrimidine substituted benzenepropanoic acid derivative, its preparation method and use in curing polycystic kidney disease SHANGHAI INST MATERIA MEDICA (CN) 2007-10-17 CN disclosed