SCHEMBL27704161

SCHEMBL27704161

O=Cc1ccc2c(c1)nnn2-c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
NPC1 O15118 2/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
ALDH1A1 P00352 5/20 0.50
ATM Q13315 2/20 0.46
FGFR1 P11362 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
DHODH Q02127 1/20 0.41
CYP2A6 P11509 1/20 0.39
P2RX7 Q99572 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
TSHR P16473 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.36
KCNMA1 Q12791 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14944391 0.83 FGFR1 (0.57) KDM4ENPC1L3MBTL1ALDH1A1ATM
SCHEMBL10357737 0.81 CA12 (0.51) KDM4ENPC1L3MBTL1ALDH1A1ATM
SCHEMBL19911581 0.76 NPC1 (1.00) KDM4ENPC1L3MBTL1ALDH1A1ATM
SCHEMBL19911612 0.76 NPC1 (0.66) KDM4ENPC1L3MBTL1ALDH1A1SMN1; SMN2
SCHEMBL9505827 0.76 NPC1 (0.66) KDM4ENPC1L3MBTL1ALDH1A1ATM
SCHEMBL18167005 0.76 KDM4E (0.66) KDM4ENPC1L3MBTL1ALDH1A1FGFR1
SCHEMBL3807006 0.76 NPC1 (0.66) KDM4ENPC1L3MBTL1ALDH1A1ATM
SCHEMBL27704159 0.75 KDM4E (0.60) KDM4ENPC1L3MBTL1ALDH1A1ATM
SCHEMBL2490016 0.75 HCAR3 (0.60) KDM4ENPC1L3MBTL1FGFR1HPGD
SCHEMBL165333 0.74 SMN1; SMN2 (0.71) KDM4ENPC1L3MBTL1ALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101193869-B Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMA 2011-03-02 CN disclosed
CN-101193869-A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMA (DE) 2008-06-04 CN disclosed