SCHEMBL27709366

SCHEMBL27709366

C=CC(c1ccc2cc(-c3ccc(F)cc3)ccc2c1)S(=O)(=O)c1ccccc1-n1ccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 5/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
FBP1 P09467 1/20 0.35
CYP19A1 P11511 6/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
CCR3 P51677 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP2C19 P33261 1/20 0.32
PMP22 Q01453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4069804 0.78 MAOA (0.40) CYP17A1MAOAMAOBFBP1CYP19A1
SCHEMBL27709365 0.74 CCR3 (0.36) CYP17A1MAOAMAOBFBP1CYP19A1
SCHEMBL27847380 0.68 IDO1 (0.40) CYP17A1FBP1CYP19A1CYP11B1CYP11B2
SCHEMBL27828854 0.68 CYP3A4 (0.41) CYP17A1FBP1CYP19A1CYP11B1CYP11B2
SCHEMBL2049363 0.64 IDO1 (0.51) CYP17A1MAOAMAOBCYP19A1CYP11B1
SCHEMBL6447916 0.62 IDO1 (0.57) FBP1MEN1KMT2AALDH1A1LMNA
SCHEMBL7186898 0.62 IDO1 (0.53) FBP1CYP19A1CYP11B1CYP11B2MEN1
SCHEMBL10592832 0.62 IDO1 (0.57) FBP1CYP19A1CYP11B1CYP11B2MEN1
SCHEMBL5800340 0.59 CYP19A1 (0.74) MAOAMAOBCYP19A1CYP11B1CYP11B2
SCHEMBL16382293 0.58 IDO1 (0.73) CYP19A1CYP11B1CYP11B2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101068776-A As 5HT2AArylsulfonyl naphthalene derivatives as antagonists MERCH SHARP & DOHME LTD (GB) 2007-11-07 CN disclosed