SCHEMBL2771304

SCHEMBL2771304

CCS(C)(c1cccc(C(=O)O)c1)c1ccc(OCc2c(C(C)C)cnn2-c2ccccc2OC(F)(F)F)cc1C

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 6/20 0.43
MRGPRX4 Q96LA9 5/20 0.35
PRKAG1 P54619 1/20 0.34
PRKAA2 P54646 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
PPARG P37231 2/20 0.34
TRPM8 Q7Z2W7 1/20 0.33
LNPEP Q9UIQ6 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PKM P14618 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PPARD Q03181 1/20 0.32
P2RY1 P47900 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2769947 0.93 NR1H4 (0.39) NR1H4TRPM8LNPEP
SCHEMBL2775280 0.91 NR1H4 (0.40) NR1H4LNPEPPPARDP2RY1
SCHEMBL2771579 0.88 NR1H4 (0.40) NR1H4TRPM8LNPEPPPARD
SCHEMBL2771162 0.84 NR1H4 (0.61) NR1H4MRGPRX4
SCHEMBL2770975 0.82 NR1H4 (0.44) NR1H4MRGPRX4PRKAG1PRKAA2PRKAB1
SCHEMBL2771301 0.81 NR1H4 (0.43) NR1H4MRGPRX4PRKAG1PRKAA2PRKAB1
SCHEMBL2772913 0.81 NR1H4 (0.62) NR1H4
SCHEMBL2771175 0.81 NR1H4 (0.44) NR1H4MRGPRX4PRKAG1PRKAA2PRKAB1
SCHEMBL2772915 0.81 NR1H4 (0.62) NR1H4
SCHEMBL2770877 0.81 NR1H4 (0.42) NR1H4PPARGLNPEPPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed