SCHEMBL27715330

SCHEMBL27715330

Nc1cncc(-c2cncc(-c3ccncc3Cl)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNC P24863 1/20 0.41
CDK8 P49336 1/20 0.41
GAA P10253 1/20 0.40
ADORA2A P29274 2/20 0.38
NQO2 P16083 1/20 0.38
ADORA2B P29275 1/20 0.38
CDK2 P24941 2/20 0.37
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
KDR P35968 3/20 0.36
GSK3B P49841 2/20 0.36
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
PRKACA P17612 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36
LATS1 O95835 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4693972 0.84 GAA (0.47) CCNCCDK8GAAADORA2ANQO2
SCHEMBL23143338 0.71 LMNA (0.42) GAACDK2CDC7ROCK2PRKCH
SCHEMBL3068958 0.71 HSP90AA1 (0.56) MKNK2
SCHEMBL25256670 0.69 GAA (0.52) CCNCCDK8GAACDK2KDR
SCHEMBL17610095 0.68 CDK2 (0.40) ADORA2ACDK2ALOX5APFEN1KDR
SCHEMBL14246417 0.68 ABL1 (0.66) CCNCCDK8GAACDK2ALOX5AP
SCHEMBL27736014 0.67 PDPK1 (0.41) ADORA2ACDK2ALOX5APFEN1KDR
SCHEMBL27715110 0.67 ALOX5AP (0.43) NQO2ADORA2BCDK2ALOX5APFEN1
SCHEMBL31301252 0.67 GSK3B (0.59) CCNCCDK8GAACDK2GSK3B
SCHEMBL3362503 0.66 HSP90AA1 (0.50) ADORA2ACDK2ALOX5APFEN1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101268064-A Pyrazine derivatives useful as adenosine receptor antagonists ALMIRALL LAB (ES) 2008-09-17 CN disclosed