SCHEMBL27716166

SCHEMBL27716166

CC([C]=O)n1cc(C(=O)N2CCN(c3ncccc3C(F)(F)F)CC2)c2ccc(Cl)cc21

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.50
RBP4 P02753 4/20 0.49
HSD11B1 P28845 4/20 0.49
TRPA1 O75762 1/20 0.49
TRPV1 Q8NER1 1/20 0.49
GAA P10253 1/20 0.46
POLB P06746 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27737070 0.81 SMN1; SMN2 (0.52)
SCHEMBL27737057 0.80 NAMPT (0.42)
SCHEMBL615642 0.80 AVPR1A (0.53) NPSR1RBP4HSD11B1TRPA1TRPV1
SCHEMBL613046 0.80 RBP4 (0.51) NPSR1RBP4HSD11B1TRPA1TRPV1
SCHEMBL615807 0.76 AVPR1A (0.63) NPSR1RBP4HSD11B1TRPA1TRPV1
SCHEMBL16690842 0.75 RBP4 (0.72) NPSR1RBP4HSD11B1TRPA1TRPV1
SCHEMBL16689591 0.74 HSD11B1 (0.59) NPSR1RBP4HSD11B1TRPA1TRPV1
SCHEMBL28775555 0.73 F10 (0.40)
SCHEMBL5457598 0.69 HDAC2 (0.45)
SCHEMBL12024747 0.68 KRAS (0.51) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101277945-A Indol-3-yl-carbonyl-piperidine and piperazine derivatives HOFFMANN LA ROCHE (CH) 2008-10-01 CN disclosed