SCHEMBL2771925

SCHEMBL2771925

Cc1cc(N)cc(-c2cc[nH]n2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
TSHR P16473 1/20 0.43
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.33
NOTUM Q6P988 1/20 0.32
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KCNH2 Q12809 1/20 0.31
METAP2 P50579 2/20 0.31
IDO1 P14902 1/20 0.31
XDH P47989 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5111323 0.91 NOTUM (0.36) ADORA2AADORA1NOTUMMEN1NPC1
SCHEMBL28478227 0.76 ERBB2 (0.30) KDM4ENPC1RAB9ATDP1
SCHEMBL28313237 0.76
SCHEMBL18051409 0.75 NOTUM (0.48) NOTUMIDO1
SCHEMBL654803 0.74 METAP2 (0.56) ALDH1A1TSHRSMN1; SMN2KDM4EMEN1
SCHEMBL3401179 0.74 IDO1 (0.56) TSHRSMN1; SMN2NOTUMKDM4ENPC1
SCHEMBL4649910 0.74 TSHR (0.39) ALDH1A1TSHRKDM4ENPC1TDP1
SCHEMBL19039332 0.73 POLB (0.36) ALDH1A1KDM4EMEN1MAPTRAB9A
SCHEMBL23815328 0.73 CYP2A6 (0.43) METAP2IDO1
SCHEMBL2765284 0.72 KMT2A (0.52) ALDH1A1SMN1; SMN2NOTUMKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2240506-A1 INHIBITORS OF IAP Genentech, Inc. (US) 2010-10-20 EP disclosed
WO-2009089502-A1 INHIBITORS OF IAP GENENTECH, INC. (US) 2009-07-16 WO disclosed