SCHEMBL27720673

SCHEMBL27720673

CC(C)(C)OC(=O)N1CCN(Cc2ccc3c(c2)cc(-c2nccc4c2C(C=O)NC4)n3C(=O)OC(C)(C)C)CC1

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 18/20 0.39
CCNK O75909 1/20 0.38
CDK12 Q9NYV4 1/20 0.38
ATR Q13535 1/20 0.37
ATRIP Q8WXE1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3159181 0.82 TBK1 (0.41) TBK1CCNKCDK12ATRATRIP
SCHEMBL3044658 0.76 ATR (0.38) TBK1ATRATRIP
SCHEMBL13291505 0.72 IDO1 (0.47) TBK1
SCHEMBL28768696 0.72 IDO1 (0.40) TBK1CCNKCDK12
SCHEMBL27700323 0.72 VEGFA (0.37) TBK1CCNKCDK12
SCHEMBL12946264 0.70 CHRM2 (0.44) TBK1CCNKCDK12
SCHEMBL3047734 0.70 VEGFA (0.40) TBK1CCNKCDK12
SCHEMBL3046667 0.70 IDO1 (0.42) TBK1CCNKCDK12
SCHEMBL5047151 0.69 TBK1 (0.40) TBK1CCNKCDK12ATRATRIP
SCHEMBL3039595 0.69 NR1H2 (0.36) TBK1ATRATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101163675-A Nitrogen-containing heterocyclic compound KYOWA HAKKO KOGYO KK (JP) 2008-04-16 CN disclosed