SCHEMBL2769946

SCHEMBL2769946

CCS(C)(c1cccc(CC(=O)O)c1)c1ccc(OCc2c(C(C)C)cnn2-c2c(Cl)cccc2Cl)cc1C

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 12/20 0.50
PPARD Q03181 5/20 0.36
FFAR1 O14842 5/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
KMT2A Q03164 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2772145 0.93 NR1H4 (0.51) NR1H4PPARDFFAR1
SCHEMBL2771162 0.90 NR1H4 (0.61) NR1H4MRGPRX4
SCHEMBL2771606 0.87 NR1H4 (0.57) NR1H4MRGPRX4
SCHEMBL3165073 0.87 NR1H4 (0.51) NR1H4PPARDFFAR1MRGPRX4KMT2A
SCHEMBL2770911 0.87 NR1H4 (0.52) NR1H4MRGPRX4KMT2A
SCHEMBL2775280 0.84 NR1H4 (0.40) NR1H4PPARDFFAR1
SCHEMBL2774998 0.83 NR1H4 (0.55) NR1H4PPARDFFAR1MRGPRX4KMT2A
SCHEMBL2788933 0.82 NR1H4 (0.53) NR1H4PPARDMRGPRX4KMT2ACYP4F2
SCHEMBL2773817 0.82 NR1H4 (0.54) NR1H4FFAR1
SCHEMBL2770534 0.81 NR1H4 (0.56) NR1H4PPARDFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed