SCHEMBL27722982

SCHEMBL27722982

Clc1cc(-c2cc[c]cc2)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
RECQL P46063 1/20 0.39
LOX P28300 1/20 0.39
LOXL3 P58215 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
CYP19A1 P11511 1/20 0.36
TRPA1 O75762 1/20 0.36
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
CDC7 O00311 1/20 0.36
ROCK2 O75116 1/20 0.36
MAP4K4 O95819 1/20 0.36
CDK2 P24941 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
GSK3B P49841 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4027001 0.84 IDO1 (0.55) IDO1CCNCCDK8RECQLLOX
SCHEMBL4672168 0.80 LMNA (0.52) IDO1CCNCCDK8RECQLLOX
SCHEMBL3500189 0.78 MAP4K4 (0.49) IDO1CCNCCDK8RECQLLOX
SCHEMBL29461217 0.78 ADORA2A (0.56) IDO1CCNCCDK8RECQLLOX
SCHEMBL2329610 0.78 ADORA2A (0.56) IDO1CCNCCDK8RECQLLOX
SCHEMBL2183379 0.77 IDO1 (0.44) IDO1CCNCCDK8RECQLLOX
SCHEMBL25070215 0.77 ADORA2A (0.54) IDO1CCNCCDK8ADORA2AADORA1
SCHEMBL28513304 0.76 IDO1 (0.39) IDO1CCNCCDK8RECQLLOX
SCHEMBL28582294 0.75 IDO1 (0.44) IDO1
SCHEMBL2156031 0.75 DYRK1A (0.56) CCNCCDK8CDC7ROCK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101193635-A Multicyclic compounds and methods of their use LEXICON GENETICS INC (US) 2008-06-04 CN claimed
CN-102395585-A Heteroaryls and their use as pi3k inhibitors MILLENNIUM PHARM INC 2012-03-28 CN disclosed
CN-101193635-A Multicyclic compounds and methods of their use LEXICON GENETICS INC (US) 2008-06-04 CN disclosed