SCHEMBL27724735

SCHEMBL27724735

OC(CF)(c1ccc2c(ccn2-c2ccc(F)cc2)c1)c1ccc(F)c2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.51
NR3C1 P04150 9/20 0.37
EPHX2 P34913 1/20 0.36
MGLL Q99685 5/20 0.36
BIRC5 O15392 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC10 Q969S8 1/20 0.32
HDAC11 Q96DB2 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
PLA2G4A P47712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28769706 0.94 KCNH2 (0.42) KCNH2NR3C1MGLLBIRC5HDAC3
SCHEMBL4283107 0.84 KCNH2 (0.52) KCNH2NR3C1MGLLBIRC5
SCHEMBL27724676 0.82 NR3C1 (0.58) NR3C1
SCHEMBL4285257 0.82 KCNH2 (0.49) KCNH2NR3C1EPHX2MGLLBIRC5
SCHEMBL27704110 0.78 NR3C1 (0.38) KCNH2NR3C1
SCHEMBL4278445 0.78 NR3C1 (0.43) KCNH2NR3C1MGLLBIRC5HDAC3
SCHEMBL28773308 0.76 KCNH2 (0.47) KCNH2MGLLBIRC5HDAC3HDAC4
SCHEMBL27704097 0.75 NR3C1 (0.50) NR3C1
SCHEMBL27724544 0.74 NR3C1 (0.47) NR3C1
SCHEMBL27724663 0.74 NR3C1 (0.53) NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101193869-A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMA (DE) 2008-06-04 CN claimed