SCHEMBL28773308

SCHEMBL28773308

OC(CF)(c1ccccc1)c1ccc2c(ccn2-c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.47
PLA2G4A P47712 1/20 0.44
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
MGLL Q99685 2/20 0.39
DHODH Q02127 2/20 0.35
ROCK2 O75116 1/20 0.35
PIM1 P11309 1/20 0.35
PIM3 Q86V86 1/20 0.35
BIRC5 O15392 1/20 0.35
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28769706 0.82 KCNH2 (0.42) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL4273650 0.80 KCNH2 (0.48) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL27724748 0.79 KCNH2 (0.57) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL27724578 0.76 NR3C1 (0.52)
SCHEMBL27724735 0.76 KCNH2 (0.51) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL24509143 0.75 KCNH2 (0.72) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL4272116 0.75 HRH1 (0.43) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL28080209 0.72 SMN1; SMN2 (0.47) KCNH2LMNACHRM4CHRM3
SCHEMBL27704252 0.71 KCNH2 (0.55) KCNH2PLA2G4AHDAC3HDAC4HDAC1
SCHEMBL27724540 0.71 L3MBTL1 (0.51) DHODHHPGDLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101193869-A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMA (DE) 2008-06-04 CN claimed
CN-101193869-B Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMA 2011-03-02 CN disclosed
CN-101193869-A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof BOEHRINGER INGELHEIM PHARMA (DE) 2008-06-04 CN disclosed