SCHEMBL2773027

SCHEMBL2773027

COC(=O)c1ccc(-c2ccccc2C(F)(F)F)c(C)c1.COC(=O)c1ccc(Br)c(C)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.60
PDK2 Q15119 5/20 0.47
S1PR1 P21453 2/20 0.42
P4HB P07237 1/20 0.41
RBP4 P02753 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
CHRNA1 P02708 1/20 0.39
CHRNG P07510 1/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
SLC6A2 P23975 1/20 0.39
CHRNB4 P30926 1/20 0.39
SLC6A4 P31645 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2776641 0.93 NOTUM (0.54) NOTUMPDK2S1PR1P4HBRBP4
SCHEMBL320542 0.85 NOTUM (0.54) NOTUMPDK2S1PR1P4HBRBP4
SCHEMBL536257 0.81 NOTUM (0.55) NOTUMPDK2P4HBRBP4MEN1
SCHEMBL10907300 0.79 NOTUM (0.66) NOTUMPDK2P4HBMEN1MAPT
SCHEMBL205089 0.79 NOTUM (0.60) NOTUMMEN1MAPTKMT2ANPC1
SCHEMBL10035005 0.79 NOTUM (0.52) NOTUMPDK2RBP4MAPTKMT2A
SCHEMBL536555 0.79 NOTUM (0.52) NOTUMPDK2P4HBRBP4AKR1C3
SCHEMBL10035257 0.78 NOTUM (0.52) NOTUMPDK2P4HBRBP4AKR1C3
SCHEMBL319915 0.78 RORC (0.52) PDK2S1PR1KMT2ATRPV1AKR1C3
SCHEMBL14925368 0.78 PDK2 (0.50) PDK2S1PR1NPSR1KMT2ATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193125-A2 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2010-06-09 EP disclosed
WO-2009043889-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2009-04-09 WO disclosed