Quinoline

Quinoline

SCHEMBL27730359

CC(=O)n1ccc2ccc(N)cc21.c1ccc2ncccc2c1

nearest known ligand 0.51

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.51
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 2/20 0.46
TP53 P04637 2/20 0.46
HSD17B10 Q99714 2/20 0.46
MAPT P10636 2/20 0.46
ATM Q13315 2/20 0.46
CASP1 P29466 2/20 0.46
HTT P42858 2/20 0.46
HSP90AA1 P07900 1/20 0.46
HSP90AB1 P08238 1/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CYP11B1 P15538 3/20 0.42
CYP11B2 P19099 3/20 0.42
PARP1 P09874 1/20 0.41
HPGD P15428 1/20 0.40
HTR3A P46098 1/20 0.39
CYP3A4 P08684 1/20 0.38
SLC22A12 Q96S37 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL27783727 0.86 NOTUM (0.71) NOTUMALDH1A1HTTTSHRCYP11B1
SCHEMBL397539 0.83 NOTUM (0.58) NOTUMALDH1A1KDM4ETP53HSD17B10
SCHEMBL11962998 0.83 NOTUM (0.58) NOTUMALDH1A1KDM4ETP53HSD17B10
Quinoline SCHEMBL27742132 0.82 NOTUM (0.48) NOTUMALDH1A1KDM4ETP53HSD17B10
Quinoline SCHEMBL28069387 0.75 PIK3CD (0.46) ALDH1A1KDM4ETP53HSD17B10MAPT
Quinoline SCHEMBL28837832 0.73 ALDH1A1 (0.69) ALDH1A1KDM4ETP53HSD17B10MAPT
Quinoline SCHEMBL28169251 0.72 ALDH1A1 (0.68) ALDH1A1KDM4ETP53HSD17B10MAPT
Quinoline SCHEMBL27635795 0.72 ALDH1A1 (0.74) ALDH1A1KDM4EMAPTCASP1HTT
SCHEMBL31200457 0.71 SLC22A12 (0.55) NOTUMCYP11B1CYP11B2PARP1SLC22A12
SCHEMBL853076 0.71 NOTUM (0.58) NOTUMALDH1A1KDM4ETP53HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101193867-A N-substituted benzimidazolyl c-Kit inhibitors and combinatorial benzimidazole libraries OSI PHARM INC (US) 2008-06-04 CN claimed
CN-101605758-A Methods of treating hepatitis C PTC THERAPEUTICS INC (US) 2009-12-16 CN disclosed
CN-101193867-A N-substituted benzimidazolyl c-Kit inhibitors and combinatorial benzimidazole libraries OSI PHARM INC (US) 2008-06-04 CN disclosed