Quinoline

Quinoline

SCHEMBL28069387

CC(C)(C)OC(=O)n1ccc2cc(N)ccc21.c1ccc2ncccc2c1

nearest known ligand 0.46

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.46
ABL1 P00519 2/20 0.46
EGFR P00533 2/20 0.46
HCK P08631 2/20 0.46
SRC P12931 2/20 0.46
KDR P35968 2/20 0.46
PIK3CA P42336 2/20 0.46
PIK3CB P42338 2/20 0.46
MTOR P42345 2/20 0.46
PIK3CG P48736 2/20 0.46
EPHB4 P54760 2/20 0.46
PRKDC P78527 2/20 0.46
PI4KB Q9UBF8 2/20 0.46
HSP90AA1 P07900 2/20 0.43
HSP90AB1 P08238 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TP53 P04637 1/20 0.43
MAPT P10636 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312329 0.85 PIK3CD (0.51) PIK3CDABL1EGFRHCKSRC
SCHEMBL22130186 0.76 PIK3CD (0.55) PIK3CDABL1EGFRHCKSRC
Quinoline SCHEMBL27730359 0.75 NOTUM (0.51) HSP90AA1HSP90AB1ALDH1A1KDM4ETP53
SCHEMBL759396 0.75 SLC22A12 (0.48) PIK3CDABL1EGFRHCKSRC
SCHEMBL29962730 0.75 SLC22A12 (0.48) PIK3CDABL1EGFRHCKSRC
SCHEMBL2003464 0.75 NR1H2 (0.45) PIK3CDABL1EGFRHCKSRC
SCHEMBL29701136 0.75 NOTUM (0.59) PIK3CDABL1EGFRHCKSRC
SCHEMBL691666 0.75 NOTUM (0.59) PIK3CDABL1EGFRHCKSRC
SCHEMBL28085950 0.73 NOTUM (0.57) PIK3CDABL1EGFRHCKSRC
SCHEMBL8877952 0.72 PARP1 (0.59) HSP90AA1HSP90AB1PARP1POLBSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104395312-B The Spirocyclic derivatives of 4,5-dihydro-pyrazolo [3,4-c] pyridin-2-ones, its preparation method and application SICHUAN HAISCO PHARMACEUTICAL CO.,LTD. (CN) 2016-04-27 CN disclosed