SCHEMBL27732142

SCHEMBL27732142

CC(=O)OCc1cc2ccc(-c3ccc(O)cc3C)cc2s1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 15/20 0.49
ESR1 P03372 14/20 0.49
HSD17B1 P14061 1/20 0.46
FGFR1 P11362 1/20 0.41
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
MIF P14174 1/20 0.34
PFKFB3 Q16875 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2084132 0.82 ESR2 (0.48) ESR2ESR1HSD17B1FGFR1
SCHEMBL498012 0.76 ESR2 (0.51) ESR2ESR1HSD17B1FGFR1
SCHEMBL27752654 0.74 ESR2 (0.59) ESR2ESR1HSD17B1FGFR1
SCHEMBL27752680 0.74 CYP1A2 (0.40) CYP1A2CYP2C19
SCHEMBL27741387 0.68 NPSR1 (0.46) ESR2ESR1HSD17B1CYP1A2CYP2C19
SCHEMBL4077781 0.68 ESR2 (1.00) ESR2ESR1HSD17B1FGFR1CYP1A2
SCHEMBL27752701 0.68 HSD17B1 (0.44) ESR2ESR1HSD17B1FGFR1
SCHEMBL11192747 0.65 ALDH1A1 (0.44) ESR2ESR1HSD17B1
SCHEMBL28661980 0.65 HSD17B1 (0.65) ESR2ESR1HSD17B1CYP1A2CYP2C19
SCHEMBL2082039 0.64 KDM4E (0.55) ESR2ESR1HSD17B1MIFPFKFB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101374834-B Compounds and methods for modulating FXR ELI LILLY AND CO. (US) 2011-12-14 CN disclosed
CN-101374834-A Compounds and methods for modulating FXR LILLY CO ELI (US) 2009-02-25 CN disclosed