SCHEMBL27733271

SCHEMBL27733271

[CH2]COc1c(C)cc(Br)cc1C

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
POLB P06746 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
FAAH O00519 2/20 0.32
BCHE P06276 2/20 0.32
ACHE P22303 2/20 0.32
SCN4A P35499 2/20 0.32
PKM P14618 1/20 0.31
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL292606 0.81 KMT2A (0.41) MEN1KMT2AKDM4EALDH1A1SCN4A
SCHEMBL941531 0.79 KMT2A (0.45) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL3355925 0.77 MEN1 (0.45) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL262332 0.77 MEN1 (0.41) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL1045003 0.76 TSHR (0.36) MEN1KMT2AALDH1A1
SCHEMBL27458128 0.76 KMT2A (0.50) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL6716155 0.76 KMT2A (0.42) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL8417929 0.74 KMT2A (0.49) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL3182203 0.74 KMT2A (0.53) MEN1KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL5591734 0.74 KMT2A (0.49) MEN1KMT2AKDM4EALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101389613-B Macrocyclic factor viia inhibitors useful as anticoagulants BRISTOL MYERS SQUIBB CO 2011-10-12 CN disclosed
CN-101389613-A Macrocyclic factor viia inhibitors useful as anticoagulants BRISTOL MYERS SQUIBB CO (US) 2009-03-18 CN disclosed