SCHEMBL2773358

SCHEMBL2773358

COC(=O)C(C#N)=C(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.42
ALDH1A1 P00352 6/20 0.40
L3MBTL1 Q9Y468 1/20 0.33
MAPK10 P53779 4/20 0.32
HPGD P15428 2/20 0.32
TSHR P16473 4/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31
CYP2C9 P11712 1/20 0.31
PKM P14618 1/20 0.31
ALOX15 P16050 1/20 0.31
LMNA P02545 1/20 0.31
THRB P10828 1/20 0.31
BLM P54132 1/20 0.31
BTK Q06187 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
PLK3 Q9H4B4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565667 0.83 IDO1 (0.41) IDO1ALDH1A1L3MBTL1MAPK10HPGD
SCHEMBL6719577 0.83 IDO1 (0.41) IDO1ALDH1A1L3MBTL1MAPK10HPGD
SCHEMBL6719581 0.83 IDO1 (0.41) IDO1ALDH1A1L3MBTL1MAPK10HPGD
SCHEMBL19071358 0.83 IDO1 (0.41) IDO1ALDH1A1L3MBTL1MAPK10TSHR
SCHEMBL22164166 0.83 IDO1 (0.41) IDO1ALDH1A1L3MBTL1MAPK10HPGD
SCHEMBL11990634 0.80 IDO1 (0.42) IDO1ALDH1A1L3MBTL1TSHRMAPT
SCHEMBL24846023 0.78 IDO1 (0.38) IDO1ALDH1A1L3MBTL1MAPK10HPGD
SCHEMBL20442156 0.78 IDO1 (0.38) IDO1ALDH1A1L3MBTL1MAPK10TSHR
SCHEMBL8956635 0.78 ALDH1A1 (0.50) IDO1ALDH1A1L3MBTL1TSHR
SCHEMBL21230245 0.76 IDO1 (0.40) IDO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10092881-B2 Permanent hydrophilic porous coatings and methods of making them BHA ALTAIR, LLC (US) 2018-10-09 US claimed
US-20090191399-A1 PERMANENT HYDROPHILIC POROUS COATINGS ONTO A SUBSTRATE AND POROUS MEMBRANES THEREOF GENERAL ELECTRIC COMPANY (US) 2009-07-30 US claimed
US-20090191398-A1 MEMBRANES COMPRISING HYDROPHILIC COATINGS GENERAL ELECTRIC COMPANY (US) 2009-07-30 US claimed
JP-8208585-A None JP disclosed
JP-2264259-A None JP disclosed
EP-4680252-A1 SYSTEM AND METHOD FOR FLUID CAPTURE GE Vernova Infrastructure Technology LLC (US) 2026-01-21 EP disclosed
EP-4680375-A1 SYSTEM AND METHOD FOR FLUID CAPTURE GE Vernova Technology GmbH (CH) 2026-01-21 EP disclosed
EP-4587158-A2 SYSTEM AND METHOD FOR FLUID CAPTURE USING A CROSS-LINKED BINDER General Electric Company (US) 2025-07-23 EP disclosed
CN-120091854-A System and method for capturing fluids using a cross-linked binder 通用电气技术有限公司 2025-06-03 CN disclosed
WO-2025071568-A1 SYSTEM AND METHOD FOR FLUID CAPTURE USING A SILICON-CONTAINING CROSS-LINKED BINDER GE INFRASTRUCTURE TECHNOLOGY LLC (US) 2025-04-03 WO disclosed
WO-2025038070-A2 SYSTEM AND METHOD FOR FLUID CAPTURE USING A CROSS-LINKED BINDER GENERAL ELECTRIC COMPANY (US) 2025-02-20 WO disclosed
EP-1107946-B1 CYCLOALKYL CARBOXYLIC ACID AMIDES, THEIR PRODUCTION AND THEIR USE AS FUNGICIDES IN AGRICULTURE BASF AG (DE) 2002-12-04 EP disclosed
US-6441044-B1 CROP PROTECTION AGENT BASF AKTIENGESELLSCHAFT (DE) 2002-08-27 US disclosed
EP-1212291-A1 CYCLOPROPANE CARBOXYLIC ACID AMIDES, THE PRODUCTION AND THE USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-06-12 EP disclosed
EP-1107946-A2 CYCLOALKYL CARBOXYLIC ACID AMIDES, THEIR PRODUCTION AND THEIR USE AS FUNGICIDES IN AGRICULTURE BASF AKTIENGESELLSCHAFT (DE) 2001-06-20 EP disclosed
WO-2001019782-A1 CYCLOPROPANE CARBOXYLIC ACID AMIDES, THE PRODUCTION AND THE USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2001-03-22 WO disclosed
EP-0990642-A1 Cycloalkylcarboxamides, their preparation and their use as fungicides BASF AKTIENGESELLSCHAFT (DE) 2000-04-05 EP disclosed
WO-2000012465-A2 CYCLOALKYL CARBOXYLIC ACID AMIDES, THEIR PRODUCTION AND THEIR USE AS FUNGICIDES IN AGRICULTURE BASF AKTIENGESELLSCHAFT (DE) 2000-03-09 WO disclosed
JP-H08208585-A PRODUCTION OF ALPHA-CYANO-TERT-BUTYLACETIC ACID LOWER ALKYL ESTER SUMITOMO CHEM CO LTD 1996-08-13 JP disclosed
JP-H02264259-A POSITIVE TYPE RESIST COMPOSITION AND PATTERN FORMING METHOD TOPPAN PRINTING CO LTD 1990-10-29 JP disclosed