SCHEMBL27733729

SCHEMBL27733729

CC(C)(C)OC(=O)[C@@]1(C)C(=O)CN(OCc2ccccc2)C1=C=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
AKT1 P31749 1/20 0.33
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CTSS P25774 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
SYK P43405 1/20 0.32
PPARA Q07869 1/20 0.32
KMT2A Q03164 1/20 0.31
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CA12 O43570 1/20 0.31
CA1 P00915 1/20 0.31
CA7 P43166 1/20 0.31
CA14 Q9ULX7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27713416 1.00 ALDH1A1 (0.40) ALDH1A1AKT1POLBCYP3A4CYP2C9
SCHEMBL27733735 0.88 ALDH1A1 (0.37) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL27713389 0.88 ALDH1A1 (0.37) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL28775111 0.86 ALDH1A1 (0.46) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL27713377 0.76 ALDH1A1 (0.42) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL27733741 0.76 ALDH1A1 (0.42) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL27733866 0.76 KMT2A (0.38) ALDH1A1AKT1CTSSL3MBTL1SYK
SCHEMBL28770888 0.76 KMT2A (0.38) ALDH1A1AKT1CTSSL3MBTL1SYK
SCHEMBL13244923 0.67 MAPK1 (0.44) KMT2AMAPK1JAK2JAK1
SCHEMBL3975093 0.67 MEN1 (0.43) ALDH1A1CYP2C19KMT2ANPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189222-B Tri-, tetra-substituted-3-aminopyrrolidine derivative DAIICHI SANKYO CO LTD 2013-01-02 CN disclosed
CN-101189222-A Tri-, tetra-substituted-3-aminopyrrolidine derivative DAIICHI SEIYAKU CO (JP) 2008-05-28 CN disclosed