SCHEMBL27733735

SCHEMBL27733735

C=C1CN(OCc2ccccc2)C(=C=O)[C@]1(C)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
STS P08842 1/20 0.34
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GPR119 Q8TDV5 2/20 0.32
CTSL P07711 1/20 0.32
AGTR2 P50052 1/20 0.32
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CTSS P25774 1/20 0.32
PRMT5 O14744 1/20 0.32
YAP1 P46937 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27713389 1.00 ALDH1A1 (0.37) ALDH1A1JAK2JAK1STSKMT2A
SCHEMBL27733729 0.88 ALDH1A1 (0.40) ALDH1A1JAK2JAK1KMT2AL3MBTL1
SCHEMBL27713416 0.88 ALDH1A1 (0.40) ALDH1A1JAK2JAK1KMT2AL3MBTL1
SCHEMBL27733741 0.87 ALDH1A1 (0.42) ALDH1A1KMT2APOLBCYP3A4CYP2C9
SCHEMBL27713377 0.87 ALDH1A1 (0.42) ALDH1A1KMT2APOLBCYP3A4CYP2C9
SCHEMBL27733866 0.83 KMT2A (0.38) ALDH1A1KMT2AL3MBTL1CTSLCTSS
SCHEMBL28770888 0.83 KMT2A (0.38) ALDH1A1KMT2AL3MBTL1CTSLCTSS
SCHEMBL28775111 0.76 ALDH1A1 (0.46) ALDH1A1POLBCYP3A4CYP2C9CYP2C19
SCHEMBL27733746 0.67 SMN1; SMN2 (0.44) KMT2AAGTR2CYP2C19RORC
SCHEMBL27733865 0.67 SMN1; SMN2 (0.44) KMT2AAGTR2CYP2C19RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101189222-B Tri-, tetra-substituted-3-aminopyrrolidine derivative DAIICHI SANKYO CO LTD 2013-01-02 CN disclosed
CN-101189222-A Tri-, tetra-substituted-3-aminopyrrolidine derivative DAIICHI SEIYAKU CO (JP) 2008-05-28 CN disclosed