SCHEMBL27733809

SCHEMBL27733809

C=CCOc1ccc(C[S+]([O-])CCC2=CC(C)(C(=O)O)CC(C(=O)O)=C2)c(C)c1

nearest known ligand 0.31

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.31
KDM4E B2RXH2 1/20 0.31
PKM P14618 1/20 0.31
ALDH1A1 P00352 2/20 0.30
ESR1 P03372 1/20 0.30
TP53 P04637 1/20 0.30
APEX1 P27695 1/20 0.30
MAPK1 P28482 1/20 0.30
ESR2 Q92731 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
KAT6A Q92794 1/20 0.30
MTNR1A P48039 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27713382 0.87 FFAR1 (0.36) POLBKDM4EALDH1A1L3MBTL1GAA
SCHEMBL27733810 0.83 POLB (0.33) POLBKDM4EPKMALDH1A1ESR1
SCHEMBL4501360 0.67 MAOA (0.35) ALDH1A1GAAHPGDMTNR1A
SCHEMBL27606816 0.65 RAB9A (0.36) POLBKDM4ETP53TDP1L3MBTL1
SCHEMBL27446644 0.64
SCHEMBL27475943 0.64
SCHEMBL28805616 0.64
SCHEMBL27794981 0.64 CYP26B1 (0.33)
SCHEMBL4606288 0.63 MAOA (0.33) ALDH1A1GAAHPGD
SCHEMBL28069778 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101208335-A Pyrazole derivatives, their manufacture and their use as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2008-06-25 CN disclosed