SCHEMBL27734876

SCHEMBL27734876

CC(=O)Oc1c(C)c(Sc2ccc(S(C)(=O)=O)cc2)n2cc(C(F)(F)F)ccc12

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.36
AKR1C3 P42330 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
PTGS2 P35354 7/20 0.35
PTGS1 P23219 1/20 0.35
CYP2C9 P11712 1/20 0.34
AKR1B1 P15121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27734882 0.83 PTGS2 (0.35) PTGDR2AKR1C3CYP11B1CYP11B2PTGS2
SCHEMBL27714461 0.83 PTGS2 (0.35) PTGDR2PTGS2PTGS1CYP2C9AKR1B1
SCHEMBL27734880 0.82 PTGDR2 (0.41) PTGDR2AKR1C3CYP11B1CYP11B2PTGS2
SCHEMBL2773692 0.80 PTGDR2 (0.58) PTGDR2AKR1C3PTGS2PTGS1CYP2C9
SCHEMBL2770081 0.79 PTGDR2 (0.46) PTGDR2PTGS2PTGS1
SCHEMBL27714354 0.71 PTGS2 (0.33) PTGDR2PTGS2PTGS1CYP2C9AKR1B1
SCHEMBL27734984 0.70 PTGDR2 (0.55) PTGDR2PTGS2PTGS1CYP2C9AKR1B1
SCHEMBL27714352 0.70 PTGDR2 (0.35) PTGDR2PTGS2CYP2C9AKR1B1
SCHEMBL27714375 0.69 PTGDR2 (0.35) PTGDR2PTGS2PTGS1
SCHEMBL27714373 0.68 PTGDR2 (0.38) PTGDR2PTGS2PTGS1CYP2C9AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101243086-A Indolizine derivatives and their use as CRTH2 antagonists ARGENTA DISCOVERY LTD (GB) 2008-08-13 CN disclosed