SCHEMBL27735005

SCHEMBL27735005

O=CC1N(c2ccccn2)CC(c2ccccn2)=NN1c1ccccc1Br

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PRKCZ Q05513 1/20 0.32
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27755569 0.89 PRKCZ (0.36) PRKCZ
SCHEMBL27735037 0.87 PRKCZ (0.35) PRKCZ
SCHEMBL27755571 0.85 GRM5 (0.33) PRKCZ
SCHEMBL27755562 0.85 FLT3 (0.34) MEN1KMT2APRKCZ
SCHEMBL27755568 0.85 GRM5 (0.34) MEN1KMT2APRKCZ
SCHEMBL27735008 0.85 CYP2A6 (0.34) PRKCZ
SCHEMBL27755589 0.84 PRKCZ (0.31) PRKCZ
SCHEMBL27735000 0.83 PRKCZ (0.34) PRKCZ
SCHEMBL27735007 0.83 SMN1; SMN2 (0.36) PRKCZ
SCHEMBL27598051 0.81 NPSR1 (0.40) MEN1KMT2APRKCZ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101486683-B Pyridazinone and triazinone compounds and their use as pharmaceutical formulations Sanitary Material R&D Management Co.,Ltd. (JP) 2011-12-21 CN disclosed
CN-101486683-A Pyridazinone and triazinone compounds and their use as pharmaceutical formulations EISAI R&D MAN CO LTD (JP) 2009-07-22 CN disclosed
CN-100473647-C Pyridazinone and triazinone compounds and their use as pharmaceutical formulations EISAI CO LTD (JP) 2009-04-01 CN disclosed