SCHEMBL27735779

SCHEMBL27735779

COc1cc(N2CCC(c3nc(C(=O)Nc4nc5ccc(C(=O)c6ccsc6)cc5[nH]4)cs3)CC2)cc(OC)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.62
NFKB2 Q00653 1/20 0.62
RELA Q04206 1/20 0.62
ALDH1A1 P00352 2/20 0.41
ABL1 P00519 2/20 0.41
LMNA P02545 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
HTT P42858 2/20 0.41
HIF1A Q16665 2/20 0.41
KDR P35968 2/20 0.41
ABCC4 O15439 1/20 0.41
USP2 O75604 1/20 0.41
TUBB4A P04350 3/20 0.40
TUBB P07437 3/20 0.40
TUBA3C P0DPH7 3/20 0.40
TUBA1B P68363 3/20 0.40
TUBA4A P68366 3/20 0.40
TUBB4B P68371 3/20 0.40
TUBB3 Q13509 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27735776 0.92 NFKB1 (0.70) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2141311 0.90 NFKB1 (0.57) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2141238 0.89 NFKB1 (0.60) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2139185 0.83 NFKB1 (0.66) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2139575 0.82 NFKB1 (0.87) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2139370 0.76 NFKB1 (1.00) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL30316128 0.76 NFKB1 (1.00) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL14046922 0.75 NFKB1 (0.71) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2140541 0.75 NFKB1 (0.61) NFKB1NFKB2RELAALDH1A1ABL1
SCHEMBL2139666 0.74 NFKB1 (0.69) NFKB1NFKB2RELAALDH1A1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101405278-A Novel heterocyclic NF-kB inhibitors 4SC AG (DE) 2009-04-08 CN disclosed