SCHEMBL27736136

SCHEMBL27736136

O=C(O)c1ccc(-c2ccccc2)c(C(=O)c2ccccc2)c1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C8 P10632 3/20 0.71
CYP2C9 P11712 2/20 0.71
KDM4E B2RXH2 1/20 0.66
ALDH1A1 P00352 2/20 0.54
SRD5A2 P31213 3/20 0.53
HCRTR1 O43613 1/20 0.53
HCRTR2 O43614 1/20 0.53
CDC25B P30305 2/20 0.53
ATM Q13315 1/20 0.53
KMO O15229 1/20 0.52
AKR1C3 P42330 1/20 0.50
SRD5A1 P18405 1/20 0.49
CDC25A P30304 1/20 0.49
HSD17B10 Q99714 1/20 0.49
TTR P02766 1/20 0.49
FOLH1 Q04609 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL594370 0.87 FOLH1 (0.59) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL22729968 0.85 TTR (0.52) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
Water SCHEMBL28745832 0.85 FOLH1 (0.57) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL29562805 0.85 TTR (0.52) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL28791455 0.84 CYP2C8 (0.50) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL5959807 0.84 CYP2C9 (0.58) CYP2C8CYP2C9ALDH1A1HCRTR1HCRTR2
SCHEMBL3104353 0.82 KDM4C (0.53) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL5215160 0.82 BCAT2 (0.61) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL28427727 0.81 KDM4E (0.89) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2
SCHEMBL29941267 0.81 KDM4E (0.89) CYP2C8CYP2C9KDM4EALDH1A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101208342-A Pyrrolobenzodiazepine * pyridine carboxamides and derivatives as follicle stimulating hormone receptor antagonists WYETH CORP (US) 2008-06-25 CN disclosed