SCHEMBL27739136

SCHEMBL27739136

Cc1cc(Br)ccc1C(N)=O.O=S(=O)(O)C=Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.43
NFE2L2 Q16236 1/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
GPR27 Q9NS67 1/20 0.41
CYP1B1 Q16678 1/20 0.40
DGAT1 O75907 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 2/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
HTT P42858 2/20 0.39
LMNA P02545 1/20 0.39
HSP90AA1 P07900 1/20 0.39
THRB P10828 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5411190 1.00 PTGS2 (0.43) PTGS2NFE2L2CA12CA9GPR27
SCHEMBL27738946 0.88 STAT3 (0.45) PTGS2NFE2L2CA12CA9ALDH1A1
SCHEMBL5423015 0.88 STAT3 (0.45) PTGS2NFE2L2CA12CA9ALDH1A1
SCHEMBL4255157 0.86 MKNK1 (0.49) PTGS2NFE2L2CYP1B1KMT2AMAPT
SCHEMBL27706028 0.86 MKNK1 (0.49) PTGS2NFE2L2CYP1B1KMT2AMAPT
SCHEMBL27738949 0.86 CA12 (0.43) CA12CA9CYP1B1DGAT1ALDH1A1
SCHEMBL5417556 0.86 CA12 (0.43) CA12CA9CYP1B1DGAT1ALDH1A1
SCHEMBL4619299 0.85 ALDH1A1 (0.45) NFE2L2ALDH1A1KMT2AMAPTSMN1; SMN2
SCHEMBL27738953 0.85 PTGS2 (0.43) PTGS2NFE2L2GPR27CYP1B1ALDH1A1
SCHEMBL5415469 0.85 PTGS2 (0.43) PTGS2NFE2L2GPR27CYP1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101268042-A Styryl sulfonamides, their preparation and use as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2008-09-17 CN claimed
CN-101268042-A Styryl sulfonamides, their preparation and use as pharmaceutical agents HOFFMANN LA ROCHE (CH) 2008-09-17 CN disclosed