SCHEMBL2774243

SCHEMBL2774243

CC(=O)Nc1c(C(=O)O)oc2ccccc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.76
ALDH1A1 P00352 2/20 0.76
KDM4E B2RXH2 3/20 0.68
HTT P42858 1/20 0.68
MAPK1 P28482 2/20 0.65
MEN1 O00255 1/20 0.65
KMT2A Q03164 1/20 0.65
HTR2C P28335 1/20 0.61
POLB P06746 3/20 0.59
TP53 P04637 2/20 0.59
SMN1; SMN2 Q16637 4/20 0.56
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C19 P33261 2/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2C9 P11712 1/20 0.56
HSD17B10 Q99714 1/20 0.56
LMNA P02545 1/20 0.53
CYP2D6 P10635 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20659868 0.86 TSHR (0.69) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL13744476 0.85 TSHR (0.72) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL4496335 0.85 ALDH1A1 (0.57) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL15714287 0.84 TSHR (0.68) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL4496337 0.84 SMN1; SMN2 (0.63) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL13744123 0.83 TSHR (0.65) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL6857800 0.81 TSHR (0.62) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL29853112 0.80 LMNA (0.62) TSHRALDH1A1KDM4EHTTPOLB
SCHEMBL18702845 0.80 TP53 (0.55) TSHRALDH1A1KDM4EHTTMAPK1
SCHEMBL2775100 0.80 TSHR (0.61) TSHRALDH1A1KDM4EHTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2161266-A1 Benzofuran derivatives as orexin receptor antagonists EVOTEC Neurosciences GmbH (DE) 2010-03-10 EP disclosed
EP-2161266-A1 Benzofuran derivatives as orexin receptor antagonists EVOTEC Neurosciences GmbH (DE) 2010-03-10 EP disclosed
EP-0187487-B1 BENZOTHIOPHENES AND BENZOFURANS HAVING ANTIALLERGIC ACTIVITY WARNER-LAMBERT COMPANY (US) 1990-08-29 EP disclosed
US-4703053-A Benzothiophenes and benzofurans and antiallergic use thereof WARNER-LAMBERT COMPANY (US) 1987-10-27 US disclosed
EP-0187487-A1 Benzothiophenes and benzofurans having antiallergic activity WARNER-LAMBERT COMPANY (US) 1986-07-16 EP disclosed