SCHEMBL27742901

SCHEMBL27742901

O=COC(Cc1c[nH]nc1C(F)(F)F)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
KCNK2 O95069 1/20 0.32
KCNH2 Q12809 1/20 0.32
CACNA1C Q13936 1/20 0.32
PARP1 P09874 1/20 0.30
GSR P00390 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27649707 0.86 PARP1 (0.32) PARP1
SCHEMBL28279524 0.82 CYP2C8 (0.32)
SCHEMBL27528515 0.81 GLS (0.32)
SCHEMBL27735924 0.81
SCHEMBL27699978 0.79
SCHEMBL28058866 0.76 IDO1 (0.33) PARP1
SCHEMBL27809350 0.76
SCHEMBL27896647 0.75 SLC6A2 (0.31) SLC6A2SLC6A4SLC6A3KCNK2KCNH2
SCHEMBL27934760 0.74
SCHEMBL27912622 0.73 GSR (0.38) SLC6A2SLC6A4GSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105722829-A Process for the regioselective synthesis of pyrazoles 伊萨格洛公司 2016-06-29 CN disclosed
CN-102993097-A Pyrazole amide compound and application thereof UNIV GUIZHOU 2013-03-27 CN disclosed
CN-101316844-A Inhibitors of diacylglycerol acyltransferase (DGAT) HOFFMANN LA ROCHE (CH) 2008-12-03 CN disclosed