SCHEMBL2774397

SCHEMBL2774397

CNCc1ccc(OCC(=O)O)c(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.57
S1PR2 O95136 1/20 0.49
S1PR1 P21453 1/20 0.49
S1PR3 Q99500 1/20 0.49
LPAR2 Q9HBW0 1/20 0.49
HSD17B10 Q99714 3/20 0.48
TSHR P16473 2/20 0.48
ALOX15 P16050 1/20 0.48
PTGDR2 Q9Y5Y4 5/20 0.48
TDP1 Q9NUW8 3/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 3/20 0.46
NPC1 O15118 1/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL989199 0.82 KMT2A (0.48) S1PR2S1PR1S1PR3LPAR2HSD17B10
SCHEMBL12988089 0.79 MEN1 (0.47) HSD17B10TSHRALOX15PTGDR2TDP1
SCHEMBL6183033 0.78 MAPT (0.51) PKMMEN1KMT2AMAPTALDH1A1
SCHEMBL3714744 0.76 PKM (0.66) PKMTSHRPTGDR2TDP1MEN1
SCHEMBL5940467 0.76 MAPT (0.64) TDP1MEN1KMT2AMAPTALDH1A1
SCHEMBL1615073 0.76 PKM (0.70) PKMTSHRPTGDR2TDP1MAPT
SCHEMBL4975454 0.75 PKM (0.64) PKMHSD17B10TSHRALOX15PTGDR2
SCHEMBL5502944 0.74 PKM (0.68) PKMHSD17B10TSHRALOX15PTGDR2
SCHEMBL2112042 0.73 PKM (1.00) PKMPTGDR2TDP1MAPTALDH1A1
SCHEMBL1369311 0.73 TDP1 (0.70) PKMTSHRPTGDR2TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010102154-A2 BIARYL OXYACETIC ACID COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-09-10 WO disclosed