SCHEMBL2774437

SCHEMBL2774437

Cc1cc(OCc2c(C)cnn2-c2c(Cl)cccc2Cl)ccc1-c1ccc(C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 9/20 0.50
MRGPRX4 Q96LA9 2/20 0.44
MAP4K4 O95819 3/20 0.40
NR4A2 P43354 1/20 0.40
RXRA P19793 2/20 0.39
RXRB P28702 2/20 0.39
RXRG P48443 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2771697 0.90 NR1H4 (0.63) NR1H4MRGPRX4
SCHEMBL2772558 0.87 NR1H4 (0.47) NR1H4MRGPRX4MAP4K4NR4A2RXRA
SCHEMBL2773781 0.84 NR1H4 (0.45) NR1H4MRGPRX4NR4A2RXRARXRB
SCHEMBL3150343 0.84 NR1H4 (0.51) NR1H4MRGPRX4NR4A2
SCHEMBL2771625 0.84 NR1H4 (0.47) NR1H4MRGPRX4RXRARXRBRXRG
SCHEMBL498129 0.83 NR1H4 (0.68) NR1H4MRGPRX4
SCHEMBL2833139 0.83 NR1H4 (0.44) NR1H4MRGPRX4NR4A2RXRARXRB
SCHEMBL2770495 0.83 NR1H4 (0.67) NR1H4MRGPRX4
SCHEMBL2772894 0.82 NR1H4 (0.67) NR1H4MRGPRX4
SCHEMBL2773617 0.82 NR1H4 (0.47) NR1H4MRGPRX4NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029547-B1 FXR AGONISTS LILLY CO ELI (US) 2010-04-28 EP disclosed